MabThera MoA
MabThera eradicates lymphoma cells via the CD20 receptor and multiple mechanisms, including complement-mediated cytotoxicity (CDC), antibody-dependent cytotoxicity (ADCC) and apoptosis.
- MabThera directly binds to the C1q complement factor, initiating complement-mediated lysis of circulating B-cells4.
- Additionally, MabThera binds strongly to Fc receptors on human effector cells, such as macrophages and natural killer cells, inducing ADCC to destroy lymphoma cells2.
- Furthermore, MabThera demonstrates an effect on the proliferation and differentiation of malignant lymphoid cells, and cell cycle regulation1,3,5,6, as well as inducing apoptosis, or programmed cell death, in vitro2.
References
- Li H, et al. J Biol Chem 2003; 278: 42427-42434.
- Maloney DG, et al. Blood (ASH Annual Meeting Abstracts) 1996; 88 (Supplement 1): abs 637a.
- Mathas S, et al. Cancer Res 2000; 60: 7170-7176.
- Reff ME, et al. Blood 1994; 83: 435-445.
- Riley JK, Sliwkowski MX. Semin Oncol 2000; 27: 17-24.
- Shan D, et al. Cancer Immunol Immunother 2000; 48: 673- 683.